zuranolone
CHEBI:CHEBI_228302
Definition
A 3-hydroxy steroid that is 5beta-19-norpregnane substituted by hydroxy, methyl, oxo, and 4-cyano-1H-pyrazol-1-yl groups at positions 3, 3, 20 and 21, respectively. It is a positive allosteric modulator of GABAA receptor developed by Sage Therapeutics and Biogen for the treatment of postpartum depression in adults.
Chemical Information
- Molecular Formula
- C25H35N3O2
- Molecular Mass
- 409.574
- Charge
- 0
- SMILES
- [H][C@@]1(CC[C@@]2([H])[C@]3([H])CC[C@]4([H])C[C@](C)(O)CC[C@]4([H])[C@@]3([H])CC[C@]12C)C(=O)CN1C=C(C=N1)C#N
- InChI
- InChI=1S/C25H35N3O2/c1-24(30)9-7-18-17(11-24)3-4-20-19(18)8-10-25(2)21(20)5-6-22(25)23(29)15-28-14-16(12-26)13-27-28/h13-14,17-22,30H,3-11,15H2,1-2H3/t17-,18+,19-,20-,21+,22-,24-,25+/m1/s1
- InChIKey
- HARRKNSQXBRBGZ-GVKWWOCJSA-N
Alternative Names
- 1-(3alpha-hydroxy-3beta-methyl-20-oxo-5beta-19-norpregnan-21-yl)-1H-pyrazole-4-carbonitrile
- 1-[(3alpha,5beta)-3-hydroxy-3-methyl-20-oxo-19-norpregnan-21-yl]-1H-pyrazole-4-carbonitrile
- BIIB-125
- BIIB125
- S-812217
- SAGE 217
- SAGE-217
- SAGE217
- SGE 797
- SGE-797
- zuranolone
- zuranolonum
- Zurzuvae
Drug Classification
-
20-oxo steroidView Class →
CHEBI:36885
-
nitrileView Class →
CHEBI:18379
-
processed material
-
3-hydroxy steroidView Class →
CHEBI:36834
-
pyrazolesView Class →
CHEBI:26410
-
t148407
-
t148529
-
t148764
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- DRON_00010000
- 2669905
- oboInOwl#hasDbXref
- Wikipedia:Zuranolone
- core#notation
- CHEBI:228302
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- has_treatment
- http://purl.obolibrary.org/obo/DOID_9478
- owl#annotatedSource
- t148800
- owl#someValuesFrom
- t4009936
- oboInOwl#hasOBONamespace
- chebi_ontology
- DRON_00010000
- 2669905
- oboInOwl#hasDbXref
- Wikipedia:Zuranolone
- oboInOwl#id
- CHEBI:228302
- core#notation
- CHEBI:228302
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_50268
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class