Edrophonium
CHEBI:CHEBI_251408
Definition
A quaternary ammonium ion that is N-ethyl-N,N-dimethylanilinium in which one of the meta positions is substituted by a hydroxy group. It is a reversible inhibitor of cholinesterase, with a rapid onset (30-60 seconds after injection) but a short duration of action (5-15 minutes). The chloride salt is used in myasthenia gravis both diagnostically and to distinguish between under- or over-treatment with other anticholinesterases. It has also been used for the reversal of neuromuscular blockade in anaesthesia, and for the management of poisoning due to tetrodotoxin, a neuromuscular blocking toxin found in puffer fish and other marine animals.
Chemical Information
- Molecular Formula
- C10H16NO
- Molecular Mass
- 166.24010
- Charge
- +1
- SMILES
- CC[N+](C)(C)c1cccc(O)c1
- InChI
- InChI=1S/C10H15NO/c1-4-11(2,3)9-6-5-7-10(12)8-9/h5-8H,4H2,1-3H3/p+1
- InChIKey
- VWLHWLSRQJQWRG-UHFFFAOYSA-O
Alternative Names
- (3-hydroxyphenyl)dimethylethylammonium
- 3-hydroxy-N,N-dimethyl-N-ethylanilinium
- edrophonium
- Edrophonium
- EDROPHONIUM
- EDROPHONIUM ION
- Ethyl-(3-hydroxy-phenyl)-dimethyl-ammonium
- N-ethyl-3-hydroxy-N,N-dimethylanilinium
- N-ethyl-3-hydroxy-N,N-dimethylbenzenaminium
Treatment Applications
-
congenital myasthenic syndrome 22View Disease →
DOID:0080587
-
congenital myasthenic syndrome 12View Disease →
DOID:0110660
-
congenital myasthenic syndrome 1BView Disease →
DOID:0110662
-
congenital myasthenic syndrome 3CView Disease →
DOID:0110664
-
congenital myasthenic syndrome 3BView Disease →
DOID:0110665
-
congenital myasthenic syndrome 13View Disease →
DOID:0110676
-
congenital myasthenic syndrome 4AView Disease →
DOID:0110678
-
neonatal myasthenia gravisView Disease →
DOID:14043
Drug Classification
-
phenolsView Class →
CHEBI:33853
-
quaternary ammonium ionView Class →
CHEBI:35267
-
t151418
-
t151590
-
t151726
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- DRON_00010000
- 3752
- oboInOwl#hasDbXref
- PMID:7488499
- core#notation
- CHEBI:251408
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- oboInOwl#hasOBONamespace
- chebi_ontology
- DRON_00010000
- 3752
- oboInOwl#hasDbXref
- PMID:7488499
- oboInOwl#id
- CHEBI:251408
- core#notation
- CHEBI:251408
- oboInOwl#hasAlternativeId
- CHEBI:4758
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_37733
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class
- rdf-schema#range
- https://w3id.org/def/predibionto#has_drug_108771
- rdf-schema#domain
- https://w3id.org/def/predibionto#has_side_effect11436
- owl#annotatedSource
- t152158
- owl#someValuesFrom
- t540655