Discuss This Drug

azelastine

CHEBI:CHEBI_2950

Definition

A phthalazine compound having an oxo substituent at the 1-position, a 1-methylazepan-4-yl group at the 2-position and a 4-chlorobenzyl substituent at the 4-position.

Chemical Information

Molecular Formula
C22H24ClN3O
Molecular Mass
381.89800
Charge
0
SMILES
CN1CCCC(CC1)n1nc(Cc2ccc(Cl)cc2)c2ccccc2c1=O
InChI
InChI=1S/C22H24ClN3O/c1-25-13-4-5-18(12-14-25)26-22(27)20-7-3-2-6-19(20)21(24-26)15-16-8-10-17(23)11-9-16/h2-3,6-11,18H,4-5,12-15H2,1H3
InChIKey
MBUVEWMHONZEQD-UHFFFAOYSA-N

Alternative Names

  • 4-(4-chlorobenzyl)-2-(1-methylazepan-4-yl)phthalazin-1(2H)-one
  • 4-(p-Chlorobenzyl)-2-(hexahydro-1-methyl-1H-azepin-4-yl)-1-(2H)-phthalazinone
  • azelastina
  • azelastine
  • azelastinum

Drug Classification

Important Medical Information

⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.

  • Always consult with a healthcare professional before starting, stopping, or modifying any medication.
  • Side effects may vary and this list may not be comprehensive.
  • Drug interactions may occur with other medications.

Additional Identifiers

core#notation
CHEBI:2950
DRON_00010000
18603
oboInOwl#hasDbXref
Wikipedia:Azelastine

Additional References

Wikipedia:Azelastine

🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.

Additional Attributes

core#notation
CHEBI:2950
listing_expiration_date
20241231
route
INTRAOCULAR
spl_id
ce1faa16-c6b2-46ea-8726-58f14737fea0
package_ndc
62991-3200-1
marketing_start_date
20120524
product_type
BULK INGREDIENT
marketing_category
BULK INGREDIENT FOR HUMAN PRESCRIPTION COMPOUNDING
dosage_form
SPRAY, METERED
labeler_name
Daito Pharmaceutical Co., Ltd
application_number
ANDA078621
product_ndc
50090-7461
oboInOwl#hasOBONamespace
chebi_ontology
DRON_00010000
18603
oboInOwl#hasDbXref
Wikipedia:Azelastine
oboInOwl#id
CHEBI:2950
generic_name
Azelastine Hydrochloride and Fluticasone Propionate
brand_name
Astepro Allergy
brand_name_base
Astepro Allergy
RO_0000087
http://purl.obolibrary.org/obo/CHEBI_37955
oboInOwl#inSubset
http://purl.obolibrary.org/obo/chebi#3_STAR
package_marketing_start_date
16-FEB-24
package_description
25 g in 1 JAR (62991-3200-1)
rxcui
1797884
active_ingredient_name
AZELASTINE HYDROCHLORIDE
active_ingredient_strength
500 g/g
unii
0L591QR10I
pharm_class
Histamine-1 Receptor Antagonist [EPC]
manufacturer_name
Somerset Therapeutics, LLC
spl_set_id
37c40f8d-269c-4df8-8ac7-cbe78f4ca5c4
upc
0370069091012
22-rdf-syntax-ns#type
http://www.w3.org/2002/07/owl#Class
has_treatment
http://purl.obolibrary.org/obo/DOID_4730
rdf-schema#domain
https://w3id.org/def/predibionto#has_side_effect15094
owl#annotatedSource
t173184
owl#someValuesFrom
t3020035