pitavastatin
CHEBI:CHEBI_32020
Definition
A dihydroxy monocarboxylic acid that is (6E)-7-[2-cyclopropyl-4-(4-fluorophenyl)quinolin-3-yl]hept-6-enoic acid in which the two hydroxy groups are located at positions 3 and 5 (the 3R,5S-stereoisomer). Used as its calcium salt for treatment of hypercholesterolemia (elevated levels of cholesterol in the blood) on patients unable to sufficiently lower their cholesterol levels by diet and exercise.
Chemical Information
- Molecular Formula
- C25H24FNO4
- Molecular Mass
- 421.46080
- Charge
- 0
- SMILES
- O[C@H](C[C@H](O)\C=C\c1c(nc2ccccc2c1-c1ccc(F)cc1)C1CC1)CC(O)=O
- InChI
- InChI=1S/C25H24FNO4/c26-17-9-7-15(8-10-17)24-20-3-1-2-4-22(20)27-25(16-5-6-16)21(24)12-11-18(28)13-19(29)14-23(30)31/h1-4,7-12,16,18-19,28-29H,5-6,13-14H2,(H,30,31)/b12-11+/t18-,19-/m1/s1
- InChIKey
- VGYFMXBACGZSIL-MCBHFWOFSA-N
Alternative Names
- (3R,5S,6E)-7-[2-cyclopropyl-4-(4-fluorophenyl)quinolin-3-yl]-3,5-dihydroxyhept-6-enoic acid
- NK 104
- NK-104
- pitavastatia
- pitavastatin
- pitavastatine
- pitavastatinum
Drug Classification
-
cyclopropanesView Class →
CHEBI:51454
-
monofluorobenzenesView Class →
CHEBI:83575
-
quinolinesView Class →
CHEBI:26513
-
dihydroxy monocarboxylic acidView Class →
CHEBI:35972
-
statin (synthetic)View Class →
CHEBI:87635
-
t183147
-
t183639
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- DRON_00010000
- 861634
- oboInOwl#hasDbXref
- Wikipedia:Pitavastatin
- core#notation
- CHEBI:32020
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- oboInOwl#hasOBONamespace
- chebi_ontology
- DRON_00010000
- 861634
- oboInOwl#hasDbXref
- Wikipedia:Pitavastatin
- oboInOwl#id
- CHEBI:32020
- core#notation
- CHEBI:32020
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_22586
- chebi#is_conjugate_acid_of
- http://purl.obolibrary.org/obo/CHEBI_71260
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class
- rdf-schema#domain
- https://w3id.org/def/predibionto#has_side_effect18325
- chebi#is_conjugate_base_of
- http://purl.obolibrary.org/obo/CHEBI_71260
- owl#annotatedSource
- t183835
- owl#someValuesFrom
- t1025081