Vandetanib
CHEBI:CHEBI_49960
Definition
A quinazoline that is 7-[(1-methylpiperidin-4-yl)methoxy]quinazoline bearing additional methoxy and 4-bromo-2-fluorophenylamino substituents at positions 6 and 4 respectively. Used for the treatment of symptomatic or progressive medullary thyroid cancer in patients with unresectable locally advanced or metastatic disease.
Chemical Information
- Molecular Formula
- C22H24BrFN4O2
- Molecular Mass
- 475.35412
- Charge
- 0
- SMILES
- COc1cc2c(Nc3ccc(Br)cc3F)ncnc2cc1OCC1CCN(C)CC1
- InChI
- InChI=1S/C22H24BrFN4O2/c1-28-7-5-14(6-8-28)12-30-21-11-19-16(10-20(21)29-2)22(26-13-25-19)27-18-4-3-15(23)9-17(18)24/h3-4,9-11,13-14H,5-8,12H2,1-2H3,(H,25,26,27)
- InChIKey
- UHTHHESEBZOYNR-UHFFFAOYSA-N
Alternative Names
- ZD 6474
- ZD6474
- 4-BROMO-2-FLUORO-N-[(4E)-6-METHOXY-7-[(1-METHYLPIPERIDIN-4-YL)METHOXY]QUINAZOLIN-4(1H)-YLIDENE]ANILINE
- N-(4-bromo-2-fluorophenyl)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4-amine
- vandetanib
- Zactima
Treatment Applications
-
cauda equina neuroendocrine tumorView Disease →
DOID:0081245
-
myxoid glioneuronal tumorView Disease →
DOID:0081285
-
pituitary cancerView Disease →
DOID:1785
-
obsolete metastasis to lymph nodeView Disease →
DOID:10437
-
abducens nerve neoplasmView Disease →
DOID:14125
-
temporal lobe neoplasmView Disease →
DOID:2135
-
hypoglossal nerve neoplasmView Disease →
DOID:3198
-
cerebellopontine angle tumorView Disease →
DOID:3200
-
sella turcica neoplasmView Disease →
DOID:3643
-
obsolete medullary carcinomaView Disease →
DOID:3974
-
obsolete metastatic meningiomaView Disease →
DOID:4582
-
obsolete relapsed meningiomaView Disease →
DOID:4585
-
rhabdoid meningiomaView Disease →
DOID:5058
-
childhood cerebellar neoplasmView Disease →
DOID:5059
-
myxopapillary ependymomaView Disease →
DOID:5075
-
epithelioid neurofibromaView Disease →
DOID:5149
-
atypical neurofibromaView Disease →
DOID:5153
-
nodular ganglioneuroblastomaView Disease →
DOID:5193
-
papillary ependymomaView Disease →
DOID:5505
-
adult papillary meningiomaView Disease →
DOID:7826
-
parapharyngeal meningiomaView Disease →
DOID:8216
-
tonsillar fossa cancerView Disease →
DOID:8969
-
pyriform sinus cancerView Disease →
DOID:9235
-
obsolete CNS metastasesView Disease →
DOID:928
Drug Classification
-
piperidinesView Class →
CHEBI:26151
-
aromatic etherView Class →
CHEBI:35618
-
organofluorine compoundView Class →
CHEBI:37143
-
quinazolinesView Class →
CHEBI:38530
-
secondary amineView Class →
CHEBI:32863
-
organobromine compoundView Class →
CHEBI:37141
-
t234367
-
t235255
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- core#notation
- CHEBI:49960
- oboInOwl#hasDbXref
- Wikipedia:Vandetanib
- DRON_00010000
- 1098413
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- oboInOwl#id
- CHEBI:49960
- core#notation
- CHEBI:49960
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class
- oboInOwl#hasOBONamespace
- chebi_ontology
- oboInOwl#hasDbXref
- Wikipedia:Vandetanib
- DRON_00010000
- 1098413
- oboInOwl#hasAlternativeId
- CHEBI:49959
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_38637
- rdf-schema#range
- https://w3id.org/def/predibionto#has_drug_113776
- owl#annotatedSource
- t235312
- has_treatment
- http://purl.obolibrary.org/obo/DOID_6174
- owl#someValuesFrom
- t1083325