Pergolide
CHEBI:CHEBI_63617
Definition
A diamine that is ergoline in which the beta-hydrogen at position 8 is replaced by a (methylthio)methyl group and the hydrogen attached to the piperidine nitrogen (position 6) is replaced by a propyl group. A dopamine D2 receptor agonist which also has D1 and D2 agonist properties, it is used as the mesylate salt in the management of Parkinson's disease, although it was withdrawn from the U.S. and Canadian markets in 2007 due to an increased risk of cardiac valve dysfunction.
Chemical Information
- Molecular Formula
- C19H26N2S
- Molecular Mass
- 314.48800
- Charge
- 0
- SMILES
- [H][C@@]12Cc3c[nH]c4cccc(c34)[C@@]1([H])C[C@@H](CSC)CN2CCC
- InChI
- InChI=1S/C19H26N2S/c1-3-7-21-11-13(12-22-2)8-16-15-5-4-6-17-19(15)14(10-20-17)9-18(16)21/h4-6,10,13,16,18,20H,3,7-9,11-12H2,1-2H3/t13-,16-,18-/m1/s1
- InChIKey
- YEHCICAEULNIGD-MZMPZRCHSA-N
Alternative Names
- (8beta)-8-[(methylsulfanyl)methyl]-6-propylergoline
- pergolida
- pergolide
- pergolidum
Treatment Applications
-
aortic valve disease 1View Disease →
DOID:0080333
-
mitral valve insufficiencyView Disease →
DOID:11502
-
pulmonary valve diseaseView Disease →
DOID:5749
-
aortic valve prolapseView Disease →
DOID:5232
Drug Classification
-
organic heterotetracyclic compoundView Class →
CHEBI:38163
-
diamineView Class →
CHEBI:23666
-
methyl sulfideView Class →
CHEBI:86315
-
t262501
-
t262631
-
t262943
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- DRON_00010000
- 8047
- oboInOwl#hasDbXref
- Wikipedia:Pergolide
- core#notation
- CHEBI:63617
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- oboInOwl#hasOBONamespace
- chebi_ontology
- DRON_00010000
- 8047
- oboInOwl#hasDbXref
- Wikipedia:Pergolide
- oboInOwl#id
- CHEBI:63617
- core#notation
- CHEBI:63617
- oboInOwl#hasAlternativeId
- CHEBI:8020
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_51065
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- chebi#is_conjugate_base_of
- http://purl.obolibrary.org/obo/CHEBI_63706
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class
- rdf-schema#range
- https://w3id.org/def/predibionto#has_drug_111819
- chebi#is_conjugate_acid_of
- http://purl.obolibrary.org/obo/CHEBI_63706
- owl#annotatedSource
- t262834
- owl#someValuesFrom
- t836056