panobinostat
CHEBI:CHEBI_85990
Definition
A hydroxamic acid obtained by formal condensation of the carboxy group of (2E)-3-[4-({[2-(2-methylindol-3-yl)ethyl]amino}methyl)phenyl]prop-2-enoic acid with the amino group of hydroxylamine. A histone deacetylase inhibitor used (as its lactate salt) in combination with bortezomib and dexamethasone for the treatment of multiple myeloma.
Chemical Information
- Molecular Formula
- C21H23N3O2
- Molecular Mass
- 349.42620
- Charge
- 0
- SMILES
- Cc1[nH]c2ccccc2c1CCNCc1ccc(\C=C\C(=O)NO)cc1
- InChI
- InChI=1S/C21H23N3O2/c1-15-18(19-4-2-3-5-20(19)23-15)12-13-22-14-17-8-6-16(7-9-17)10-11-21(25)24-26/h2-11,22-23,26H,12-14H2,1H3,(H,24,25)/b11-10+
- InChIKey
- FPOHNWQLNRZRFC-ZHACJKMWSA-N
Alternative Names
- (2E)-N-hydroxy-3-[4-({[2-(2-methyl-1H-indol-3-yl)ethyl]amino}methyl)phenyl]prop-2-enamide
- LBH 589
- LBH589
- panobinostat
Treatment Applications
-
extramedullary plasmacytomaView Disease →
DOID:3720
Drug Classification
-
secondary amino compoundView Class →
CHEBI:50995
-
cinnamamidesView Class →
CHEBI:23247
-
methylindoleView Class →
CHEBI:38460
-
hydroxamic acidView Class →
CHEBI:24650
-
t309703
-
t310527
-
t310577
-
t310684
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- DRON_00010000
- 1603350
- oboInOwl#hasDbXref
- Wikipedia:Panobinostat
- core#notation
- CHEBI:85990
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- has_treatment
- http://purl.obolibrary.org/obo/DOID_5789
- rdf-schema#range
- https://w3id.org/def/predibionto#has_drug_110489
- rdf-schema#domain
- https://w3id.org/def/predibionto#has_side_effect37233
- chebi#is_conjugate_acid_of
- http://purl.obolibrary.org/obo/CHEBI_85992
- owl#annotatedSource
- t310946
- owl#someValuesFrom
- t2909181
- oboInOwl#hasOBONamespace
- chebi_ontology
- DRON_00010000
- 1603350
- oboInOwl#hasDbXref
- Wikipedia:Panobinostat
- oboInOwl#id
- CHEBI:85990
- core#notation
- CHEBI:85990
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_61115
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- chebi#is_conjugate_base_of
- http://purl.obolibrary.org/obo/CHEBI_85992
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class