alectinib
CHEBI:CHEBI_90936
Definition
An organic heterotetracyclic compound that is 6,6-dimethyl-5,6-dihydro-11H-benzo[b]carbazol-11-one carrying additional cyano, 4-(morpholin-4-yl)piperidin-1-yl and ethyl substituents at positions 3, 8 and 9 respectively. Used (as the hydrochloride salt) for the treatment of patients with anaplastic lymphoma kinase-positive, metastatic non-small cell lung cancer.
Chemical Information
- Molecular Formula
- C30H34N4O2
- Molecular Mass
- 482.618
- Charge
- 0
- SMILES
- C1OCCN(C1)C2CCN(CC2)C3=CC4=C(C=C3CC)C(C5=C(C4(C)C)NC=6C5=CC=C(C6)C#N)=O
- InChI
- InChI=1S/C30H34N4O2/c1-4-20-16-23-24(17-26(20)34-9-7-21(8-10-34)33-11-13-36-14-12-33)30(2,3)29-27(28(23)35)22-6-5-19(18-31)15-25(22)32-29/h5-6,15-17,21,32H,4,7-14H2,1-3H3
- InChIKey
- KDGFLJKFZUIJMX-UHFFFAOYSA-N
Alternative Names
- 9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5H-benzo[b]carbazole-3-carbonitrile
- AF 802
- AF-802
- alectinib
- CH 5424802
- CH5424802
Treatment Applications
-
hilar lung neoplasmView Disease →
DOID:5767
-
lung lymphomaView Disease →
DOID:6760
-
hilar lung carcinomaView Disease →
DOID:8207
Drug Classification
-
nitrileView Class →
CHEBI:18379
-
morpholinesView Class →
CHEBI:38785
-
piperidinesView Class →
CHEBI:26151
-
organic heterotetracyclic compoundView Class →
CHEBI:38163
-
aromatic ketoneView Class →
CHEBI:76224
-
t316838
-
t317291
-
t317491
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- DRON_00010000
- 1727455
- oboInOwl#hasDbXref
- Wikipedia:Alectinib
- core#notation
- CHEBI:90936
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- oboInOwl#hasOBONamespace
- chebi_ontology
- DRON_00010000
- 1727455
- oboInOwl#hasDbXref
- Wikipedia:Alectinib
- oboInOwl#id
- CHEBI:90936
- core#notation
- CHEBI:90936
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_62434
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- chebi#is_conjugate_base_of
- http://purl.obolibrary.org/obo/CHEBI_90937
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class
- has_treatment
- http://purl.obolibrary.org/obo/DOID_3908
- rdf-schema#range
- https://w3id.org/def/predibionto#has_drug_113087
- rdf-schema#domain
- https://w3id.org/def/predibionto#has_side_effect38148
- chebi#is_conjugate_acid_of
- http://purl.obolibrary.org/obo/CHEBI_90937
- owl#annotatedSource
- t317811
- owl#someValuesFrom
- t2911048