Ketotifen
CHEBI:CHEBI_92511
Definition
An organic heterotricyclic compound that is 4,9-dihydro-10H-benzo[4,5]cyclohepta[1,2-b]thiophen-10-one which is substituted at position 4 by a 1-methylpiperidin-4-ylidene group. A blocker of histamine H1 receptors with a stabilising action on mast cells, it is used (usually as its hydrogen fumarate salt) for the treatment of asthma, where it may take several weeks to exert its full effect.
Chemical Information
- Molecular Formula
- C19H19NOS
- Molecular Mass
- 309.427
- Charge
- 0
- SMILES
- CN1CCC(=C2C3=C(C(=O)CC4=CC=CC=C42)SC=C3)CC1
- InChI
- InChI=1S/C19H19NOS/c1-20-9-6-13(7-10-20)18-15-5-3-2-4-14(15)12-17(21)19-16(18)8-11-22-19/h2-5,8,11H,6-7,9-10,12H2,1H3
- InChIKey
- ZCVMWBYGMWKGHF-UHFFFAOYSA-N
Alternative Names
- 10-(1-methyl-4-piperidinylidene)-5H-benzo[1,2]cyclohepta[3,4-b]thiophen-4-one
- 4-(1-methylpiperidin-4-ylidene)-4,9-dihydro-10H-benzo[4,5]cyclohepta[1,2-b]thiophen-10-one
- ketotifen
- ketotifene
- ketotifeno
- ketotifenum
Drug Classification
-
olefinic compoundView Class →
CHEBI:78840
-
piperidinesView Class →
CHEBI:26151
-
cyclic ketoneView Class →
CHEBI:3992
-
tertiary amino compoundView Class →
CHEBI:50996
-
organic heterotricyclic compoundView Class →
CHEBI:26979
-
organosulfur heterocyclic compoundView Class →
CHEBI:38106
-
t320422
-
t320447
-
t321106
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- DRON_00010000
- 6146
- oboInOwl#hasDbXref
- Wikipedia:Ketotifen
- core#notation
- CHEBI:92511
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- oboInOwl#hasOBONamespace
- chebi_ontology
- DRON_00010000
- 6146
- oboInOwl#hasDbXref
- Wikipedia:Ketotifen
- oboInOwl#id
- CHEBI:92511
- core#notation
- CHEBI:92511
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_37955
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- chebi#is_conjugate_base_of
- http://purl.obolibrary.org/obo/CHEBI_140417
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class
- has_treatment
- http://purl.obolibrary.org/obo/DOID_4660
- chebi#is_conjugate_acid_of
- http://purl.obolibrary.org/obo/CHEBI_140417
- owl#someValuesFrom
- t3879746
- owl#annotatedSource
- t321276