exemestane
CHEBI:CHEBI_4953
Definition
A 17-oxo steroid that is androsta-1,4-diene-3,17-dione in which the hydrogens at position 6 are replaced by a double bond to a methylene group. A selective inhibitor of the aromatase (oestrogen synthase) system, it is used in the treatment of advanced breast cancer.
Chemical Information
- Molecular Formula
- C20H24O2
- Molecular Mass
- 296.40340
- Charge
- 0
- SMILES
- [H][C@@]12CC(=C)C3=CC(=O)C=C[C@]3(C)[C@@]1([H])CC[C@]1(C)C(=O)CC[C@@]21[H]
- InChI
- InChI=1S/C20H24O2/c1-12-10-14-15-4-5-18(22)20(15,3)9-7-16(14)19(2)8-6-13(21)11-17(12)19/h6,8,11,14-16H,1,4-5,7,9-10H2,2-3H3/t14-,15-,16-,19+,20-/m0/s1
- InChIKey
- BFYIZQONLCFLEV-DAELLWKTSA-N
Alternative Names
- 6-methyleneandrosta-1,4-diene-3,17-dione
- 6-methylideneandrosta-1,4-diene-3,17-dione
- exemestane
- Exemestane
- exemestano
- exemestanum
Treatment Applications
-
female breast cancerView Disease →
DOID:0050671
-
breast lobular carcinomaView Disease →
DOID:0050938
-
ductal carcinoma in situView Disease →
DOID:0060074
-
triple-receptor negative breast cancerView Disease →
DOID:0060081
-
luminal breast carcinoma AView Disease →
DOID:0060548
-
luminal breast carcinoma BView Disease →
DOID:0080674
-
aromatase excess syndromeView Disease →
DOID:0090122
-
breast cancerView Disease →
DOID:1612
-
breast cystView Disease →
DOID:10350
-
female breast central part cancerView Disease →
DOID:13799
-
breast fibroadenomaView Disease →
DOID:1618
-
breast adenomyoepitheliomaView Disease →
DOID:1642
-
invasive ductal carcinomaView Disease →
DOID:3008
-
breast granular cell tumorView Disease →
DOID:3011
-
invasive lobular carcinomaView Disease →
DOID:3457
-
obsolete breast hamartomaView Disease →
DOID:3461
-
breast metaplastic carcinomaView Disease →
DOID:4680
-
breast hemangiomaView Disease →
DOID:476
-
breast hemangiopericytomaView Disease →
DOID:5370
-
breast medullary carcinomaView Disease →
DOID:5605
-
cribriform carcinomaView Disease →
DOID:5675
-
acinic cell breast carcinomaView Disease →
DOID:5743
-
sebaceous breast carcinomaView Disease →
DOID:5760
-
breast fibrosarcomaView Disease →
DOID:6001
-
breast apocrine carcinomaView Disease →
DOID:6581
-
breast oncocytic carcinomaView Disease →
DOID:6585
-
breast juvenile papillomatosisView Disease →
DOID:6641
-
bilateral breast cancerView Disease →
DOID:6741
-
flat ductal epithelial atypiaView Disease →
DOID:6841
-
breast giant fibroadenomaView Disease →
DOID:7223
-
breast apocrine adenomaView Disease →
DOID:7540
-
breast osteosarcomaView Disease →
DOID:7787
-
female breast carcinomaView Disease →
DOID:7843
-
obsolete breast adenohibernomaView Disease →
DOID:7892
-
sporadic breast cancerView Disease →
DOID:8029
-
benign mammary dysplasiaView Disease →
DOID:9504
Drug Classification
-
17-oxo steroidView Class →
CHEBI:19168
-
3-oxo-Delta(1),Delta(4)-steroidView Class →
CHEBI:77166
-
t234500
-
t234590
-
t234665
-
t234722
-
t234765
Important Medical Information
⚕️ This information is sourced from ChEBI (Chemical Entities of Biological Interest) database and is intended for educational purposes only.
- Always consult with a healthcare professional before starting, stopping, or modifying any medication.
- Side effects may vary and this list may not be comprehensive.
- Drug interactions may occur with other medications.
Additional Identifiers
- DRON_00010000
- 258494
- oboInOwl#hasDbXref
- Wikipedia:Exemestane
- core#notation
- CHEBI:4953
Additional References
🔍 Click on any linked disease name to learn more about the conditions this medication is used to treat, or explore related drug classifications for more information about similar medications.
Additional Attributes
- oboInOwl#hasOBONamespace
- chebi_ontology
- DRON_00010000
- 258494
- oboInOwl#hasDbXref
- Wikipedia:Exemestane
- oboInOwl#id
- CHEBI:4953
- core#notation
- CHEBI:4953
- RO_0000087
- http://purl.obolibrary.org/obo/CHEBI_50790
- oboInOwl#inSubset
- http://purl.obolibrary.org/obo/chebi#3_STAR
- chebi#has_parent_hydride
- http://purl.obolibrary.org/obo/CHEBI_35509
- 22-rdf-syntax-ns#type
- http://www.w3.org/2002/07/owl#Class
- has_treatment
- http://purl.obolibrary.org/obo/DOID_5310
- rdf-schema#domain
- https://w3id.org/def/predibionto#has_side_effect26485
- owl#annotatedSource
- t235270
- owl#someValuesFrom
- t824303
- rdf-schema#range
- https://w3id.org/def/predibionto#has_drug_113802